AprinEase
Liquefied Topical Analgesic
Superior Pain Relief
Do you suffer with aches and pains of sports injuries, low back discomfort, muscle strain, or joint pain?
Normal oral pain killers and anti-inflammatories can take hours to take effect, and are diluted through your whole body. Worse yet, many can give you an upset stomach or other side effects. Most topical products just mask the pain, making the area feel cold or hot.
Now there is an alternative!
AprinEase is a topical pain reliever and anti-inflamatory that works in seconds to stop your pain, right where it hurts. Just spray it on, and the pain is gone.
AprinEase contains Triethanolamine Salicylate (TES), an anti-inflamatory found in oral pain relievers. It also contains Emu Oil and Methyl Sulfonyl Methane (MSM) using a special, proprietary formula.
Direct Application To Pain
The great news from this exciting new development in using an analgesic in this manner is that the effectiveness of the drug is wholly unimparied by using it in an external application. In fact, since the entire strength of the pain relief is concentrated on the point of pain, it is much more effective than being diluted in the body, as it is when taken orally.
Other products on the market that are used for topical pain relief either warm or cool the distressed area with camphor or menthol additives. This is simply disguising the pain -- not relieving it. They contain no analgesic. They have no transdermal effect.
Benefits of Topical Analgesics
Topical delivery offers advantages over oral administration:
1) Use smaller amounts of active ingredients
2) Avoid liver metabolism
3) Avoid degradation of active ingredients in the g. i. tract
4) No stomach upset
Delivery System of the Future
Doctors around the world are calling topicals "the delivery system of the future." It has been discovered that a high absorption rate of many
NSAIDs and pain-alleviating herbal extracts can be achieved when delivered through the skin.
While your skin acts as a barrier to water-soluble applications,
fats have been proven to pass through the skin and carry pain relief to inflamed soft tissue, such as muscle, ligament, and tendon.
Under Your Skin
The first layer of skin [epidermis] consists of laminated layers of epithelial cells which slows the evaporation of water from the inside. Its surface [stratum corneum] is a network
of furrows of different sizes.
Under the epidermis is the thickest layers of skin [dermis] which are rich in sebaceous and sweat glands, fat cells, lymph, blood vessels
and nerves.
Factors Affecting Skin Penetration
1) Oil solubility: the more oil soluble [lipophilic] the substance, the greater the skin penetration.
2) The lower the molecular weight the smaller the molecule.
3) Creams, gels and liquids penetrate better than solids.
4) Penetration enhancers improve topical absorption of lipophilic
substances.
95% Delivery
Studies have shown that when NSAIDs and nutrients are taken orally, as little as 5% make it to the area of inflammation where they are needed.
This is because of the stomach, liver and digestive system re-arranging and discarding much of them.
Summary
Our proprietary "Patch Free" liquid base technology offers a safer, quick-acting,
and easier-to-comply alternative to capsules and tablets.
References
J Pharm Sci "Linear relationships between lipophilic character and biological activity of drugs."1972 Jan;61(1):1-19
Targeted drug delivery to the skin and deeper tissues: role of physiology, solute structure and disease.Clin Exp Pharmacol Physiol 1997 Nov;24(11):874-9
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AprinEasetm
Liquefied Topical Analgesic
Indications: Mode of Action: Reduces tissue concentration of prostaglandins (hormones which produce inflammation and pain).
Uses: Treatment for joint pain, stiffness, inflammation and swelling, and aches and pains associated with arthritis and gout.
Contraindications: Do not use if you are allergic to aspirin or any non-steroidal, anti-inflammatory drug.
Warnings: For exterior skin application only and NOT to be taken orally. If your symptoms do NOT improve within 7 days or
if they get worse seek immediate medical advice. Do NOT apply to broken skin or burns or into your eyes. If this happens wash with clean cold water and seek
immediate medical advice. Not intended to reduce fever nor to treat headaches.
Precautions:
Pregnancy: Decide with your doctor whether drug benefits justify risk to unborn child.
Breast-feeding: May harm child. Avoid.
Infants & children: Not recommended for anyone younger than 15. Use only under medical supervision
Dosage: Apply liberally to the painful area, gently massaging it into the skin until absorbed, 3 or 4 times daily.
Ingredients:
Active Ingredient: Triethanolamine Salicylate 12%
Inactive Ingredients: Isopropyl Alcohol, Glycerin, Emu Oil, and Methylsulfonylmethane (MSM).
Availability: 4 oz. pump spray.
$16.95 / $11.95 for 5 or more
Order Now!
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